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Ro 60-0175
CAS No. 169675-08-5
Ro 60-0175 ( Ro 600175 )
产品货号. M12587 CAS No. 169675-08-5
Ro 60-0175 is a potent, selective 5-HT2C receptor agonist.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥2130 | 有现货 |
|
| 10MG | ￥3418 | 有现货 |
|
| 25MG | ￥5581 | 有现货 |
|
| 50MG | ￥7946 | 有现货 |
|
| 100MG | ￥10935 | 有现货 |
|
| 500MG | ￥21708 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Ro 60-0175
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Ro 60-0175 is a potent, selective 5-HT2C receptor agonist.
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产品描述Ro 60-0175 is a potent, selective 5-HT2C receptor agonist with pKi of 9, 7.5, 5.4, 5.2 and 5.6 for human 5-HT2C, 2A, 1A, 6 and 7 receptors respectively; induces hypolocomotion in rats at doses greater than 0.5 mg/kg s.c.; (0.3 and 1 mg/kg s.c.) simultaneously reduces both unpunished and punished lever pressing, a profile consistent with sedation, induces sedative-like responses via 5-HT(2C) receptor activation in vivo.
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同义词Ro 600175
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体5-HT Receptor
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研究领域——
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适应症——
化学信息
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CAS Number169675-08-5
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分子量226.68
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分子式C11H12ClFN2
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纯度>98% (HPLC)
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溶解度——
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SMILESCC(CN1C=CC2=CC(=C(C=C21)Cl)F)N.C(=CC(=O)O)C(=O)O
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化学全称1H-Indole-1-ethanamine, 6-chloro-5-fluoro-α-methyl-, (S)-
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Damjanoska KJ, et al. J Pharmacol Exp Ther. 2003 Mar;304(3):1209-16.
2. Vickers SP, et al. Br J Pharmacol. 2000 Jul;130(6):1305-14.
3. Kennett G, et al. Eur J Pharmacol. 2000 Jan 10;387(2):197-204.
4. Jenck F, et al. Eur Neuropsychopharmacol. 1998 Aug;8(3):161-8.
2. Vickers SP, et al. Br J Pharmacol. 2000 Jul;130(6):1305-14.
3. Kennett G, et al. Eur J Pharmacol. 2000 Jan 10;387(2):197-204.
4. Jenck F, et al. Eur Neuropsychopharmacol. 1998 Aug;8(3):161-8.
产品手册
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